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Updated: Aug 11, 2026

Using an α-Bungarotoxin Binding Site Tag to Study GABA A Receptor Membrane Localization and Trafficking
11:57

Using an α-Bungarotoxin Binding Site Tag to Study GABA A Receptor Membrane Localization and Trafficking

Published on: March 28, 2014

GABA(B) auto- versus hetero-receptor sensitivity: implications for novel pharmacotherapy

B Yu1, K Yamada, J P Gallagher

  • 1Department of Pharmacology and Toxicology, University of Texas Medical Branch, Galveston 77555-1031, USA.

Neuropharmacology
|December 10, 1999
PubMed
Summary

The GABA(B) agonist CGP44533 is less effective at inhibiting glutamate release than GABA release. This suggests different sensitivities of GABA and glutamate neurons to this drug.

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