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A new class of highly cytotoxic diketopiperazines

D L Boger¹, B E Fink, M P Hedrick

¹Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, La Jolla, CA 92037, USA. boger@scripps.edu

Bioorganic & Medicinal Chemistry Letters

|June 8, 2000

Abstract:

The discovery of a novel class of diketopiperazines possessing potent cytotoxic activity is described.

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