Cyclosporin A inhibits cardiac hypertrophy and enhances cardiac dysfunction during postinfarction failure in rats

E Oie1, R Bjørnerheim, O P Clausen

  • 1Merck Sharp & Dohme Cardiovascular Research Center, National Hospital, University of Oslo, Norway.

Insights

Cyclosporin A (CsA) inhibits calcineurin, reducing myocardial hypertrophy in heart failure rats. However, this inhibition worsened cardiac remodeling and function, highlighting calcineurin

Area of Science:

  • Cardiovascular Physiology
  • Molecular Cardiology
  • Pharmacology

Background:

  • Calcineurin mediates intracellular calcium signaling to myocardial hypertrophy.
  • Congestive heart failure (CHF) involves complex cardiac remodeling.
  • Calcineurin inhibitors like Cyclosporin A (CsA) impact cardiac pathways.

Purpose of the Study:

  • To investigate the effects of CsA on myocardial hypertrophy and remodeling in a rat model of CHF.
  • To elucidate the role of calcineurin-dependent pathways in compensatory cardiac hypertrophy during heart failure.

Main Methods:

  • Rats underwent left coronary artery ligation to induce CHF.
  • Rats were randomized to receive CsA or vehicle for 14 days.
  • Cardiac hypertrophy, gene expression, ventricular remodeling, and cardiac function were assessed.

Main Results:

  • CsA significantly attenuated myocardial hypertrophy and reduced skeletal alpha-actin gene expression in CHF rats.
  • CsA treatment led to increased left ventricular (LV) dilatation and reduced LV function (fractional shortening, pressure derivatives).
  • Plasma renin and endothelin-1 levels increased in CsA-treated CHF rats, indicating aggravated cardiac function.

Conclusions:

  • Calcineurin plays a critical role in compensatory myocardial hypertrophy during CHF.
  • Inhibiting compensatory hypertrophy with CsA has detrimental effects on cardiac remodeling and function post-myocardial infarction.
  • Targeting calcineurin pathways requires careful consideration due to potential adverse effects on cardiac function.

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