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Fentanyl versus sufentanil: plasma concentrations during continuous epidural postoperative infusion in children

C Lejus1, D Schwoerer, I Furic

  • 1Department of Anaesthesiology, Hôtel-Dieu, CHR Nantes, France.

Insights

This study measured plasma concentrations of fentanyl and sufentanil in children receiving epidural administration. Maximum drug levels were achieved quickly after loading doses and remained stable during continuous infusion.

Area of Science:

  • Pediatric Anesthesiology
  • Pharmacokinetics
  • Pain Management

Background:

  • Limited pharmacokinetic data exists for epidural fentanyl and sufentanil in pediatric patients.
  • Epidural analgesia is crucial for post-operative pain management in children.

Purpose of the Study:

  • To determine plasma concentrations of fentanyl and sufentanil during epidural administration in children.
  • To evaluate the pharmacokinetics of epidural opioids in pediatric surgical patients.

Main Methods:

  • Double-blind randomized study involving 12 children aged 5-12 years.
  • Administration of epidural loading doses and continuous infusions of fentanyl or sufentanil with bupivacaine.
  • Utilized an epidural patient-controlled analgesia (PCA) system for bolus doses.

Main Results:

  • Maximal median plasma concentrations for fentanyl ranged from 0.117-0.247 ng/mL.
  • Maximal median plasma concentrations for sufentanil ranged from 0.027-0.074 ng/mL.
  • Peak drug levels were reached approximately 30 minutes (fentanyl) and 20 minutes (sufentanil) after loading doses, remaining stable over 48 hours.

Conclusions:

  • Epidural fentanyl and sufentanil achieve predictable plasma concentrations in children during continuous infusion and PCA.
  • The findings provide essential pharmacokinetic data for optimizing epidural opioid analgesia in pediatric populations.

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