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Updated: Oct 8, 2026

Quantifying Agonist Activity at G Protein-coupled Receptors
11:45

Quantifying Agonist Activity at G Protein-coupled Receptors

Published on: December 26, 2011

The relative importance of the time-course of receptor occupancy and response decay on apparent antagonist potency in

M Corsi1, T Kenakin

  • 1Pharmacology Department, Glaxo Wellcome S.p.A., Verona, Italy.

Journal of Autonomic Pharmacology
|March 22, 2001
PubMed

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