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Synthesis of substituted imidazopyrazines as ligands for the human somatostatin receptor subtype 5
M O Contour-Galéra1, L Poitout, C Moinet
1Institut Henri Beaufour, Les Ulis, France. m-odile.galcera.contour@beaufour-ipsen.com
Bioorganic & Medicinal Chemistry Letters
|March 27, 2001
Abstract:
A new preparation of trisubstituted imidazopyrazines and dihydroimidazopyrazines via parallel synthesis using aminoacids and bromoketones resulted in the discovery of non-peptidic sst5 selective agonists.