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Preparation of N-(2-alkoxyvinyl)sulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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An improved synthesis of 1,2,4-oxadiazoles on solid support

K D Rice1, J M Nuss

  • 1Department of Medicinal Chemistry, Exelixis, Inc., South San Francisco, CA 94083-0511, USA. krice@exelixis.com

Bioorganic & Medicinal Chemistry Letters
|March 30, 2001
PubMed

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