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Drug-induced Sensitization of Adenylyl Cyclase: Assay Streamlining and Miniaturization for Small Molecule and siRNA Screening Applications
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Synthesis and use of FSCPX, an irreversible adenosine A1 antagonist, as a 'receptor knock-down' tool

J E van Muijlwijk-Koezen1, H Timmerman, R P van der Sluis

  • 1Leiden/Amsterdam Center for Drug Research, Department of Pharmacochemistry, Vrije Universiteit, Amsterdam, The Netherlands. muylwyk@chem.vu.nl

Bioorganic & Medicinal Chemistry Letters
|March 30, 2001
PubMed

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