Tyrosine kinase receptor activation inhibits NPR-C in lung arterial smooth muscle cells

J Z Sun1, S Oparil, P Lucchesi

  • 1Vascular Biology and Hypertension Program, Division of Cardiovascular Disease, Department of Medicine, University of Alabama at Birmingham, Birmingham, Alabama 35294, USA.

Insights

Hypoxia-responsive growth factors, fibroblast growth factors (FGF-1, FGF-2), and platelet-derived growth factor-BB (PDGF-BB) reduce atrial natriuretic peptide clearance receptor (NPR-C) expression in pulmonary arterial smooth muscle cells. This occurs via tyrosine kinase receptor activation, independent of oxygen levels.

Area of Science:

  • Pulmonary hypertension research
  • Cellular signaling pathways
  • Cardiovascular research

Background:

  • Atrial natriuretic peptide clearance receptor (NPR-C) expression is reduced in lung tissue under hypoxic conditions.
  • Pulmonary arterial smooth muscle cells (PASMCs) are key in regulating pulmonary vascular tone and remodeling.

Purpose of the Study:

  • To investigate if hypoxia-responsive growth factors (FGF-1, FGF-2, PDGF-BB) reduce NPR-C expression in PASMCs.
  • To determine if this reduction is mediated by tyrosine kinase receptors and independent of environmental oxygen tension.

Main Methods:

  • Rat PASMCs were cultured and treated with FGF-1, FGF-2, PDGF-BB, ANG II, ET-1, ANP, SNP, or cGMP under varying oxygen tensions.
  • NPR-C mRNA levels were quantified using Northern blot analysis.
  • Inhibitors of FGF receptor tyrosine kinase and MAPK pathways were used to elucidate signaling mechanisms.

Main Results:

  • FGF-1, FGF-2, and PDGF-BB significantly reduced NPR-C mRNA levels in PASMCs in a dose- and time-dependent manner.
  • Hypoxia itself, ANG II, ET-1, ANP, SNP, or cGMP did not decrease NPR-C mRNA levels.
  • The inhibitory effect of FGFs and PDGF-BB on NPR-C expression was blocked by tyrosine kinase and MAPK pathway inhibitors.

Conclusions:

  • Activation of tyrosine kinase receptors by FGF-1, FGF-2, and PDGF-BB inhibits NPR-C gene expression in PASMCs.
  • This mechanism is independent of direct hypoxic effects or G protein-coupled receptor activation.
  • These growth factors may mediate the link between hypoxia and altered NPR-C expression in the lung.

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