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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones

Published on: February 7, 2019

Synthesis of a novel C-10 spiro-epoxide of paclitaxel

M A Walker1, T D Johnson, S Huang

  • 1Bristol-Myers Squibb, Pharmaceutical Research Institute, Richard L. Gelb Center for Pharmaceutical Research and Development, 5 Research Parkway, 06492, Wallingford, CT, USA. michael.a.walker@bms.com

Bioorganic & Medicinal Chemistry Letters
|June 27, 2001
PubMed

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