Na(+)/H(+) exchange subtype 1 inhibition reduces endothelial dysfunction in vessels from stunned myocardium

J D Symons1, S Schaefer

  • 1Division of Cardiovascular Medicine, Department of Internal Medicine, University of California, Davis 95616, USA. jdsymons@ucdavis.edu

Insights

Inhibiting the Na(+)/H(+) exchanger subtype 1 (NHE(1)) with cariporide lessened ischemia-induced microvascular dysfunction in rats. However, NHE(1) inhibition did not improve myocardial contractile function after reperfusion injury.

Area of Science:

  • Cardiovascular Physiology
  • Cellular Signaling
  • Pharmacology

Background:

  • Myocardial ischemia and reperfusion induce cellular dysfunction, known as stunning.
  • The Na(+)/H(+) exchanger subtype 1 (NHE(1)) plays a role in cellular response to ischemia.
  • Understanding NHE(1) inhibition's effect on myocardial and microvascular stunning is crucial for therapeutic development.

Purpose of the Study:

  • To investigate the hypothesis that inhibiting NHE(1) during ischemia and reperfusion limits myocardial and coronary microvascular stunning.
  • To assess the impact of cariporide, an NHE(1) inhibitor, on cardiac function and resistance artery reactivity post-ischemia.

Main Methods:

  • Anesthetized rats underwent 2 x 10-min coronary artery occlusions with 5-min reperfusion, followed by 15 or 60 min of reperfusion.
  • Vehicle or cariporide was administered 15 minutes before ischemia and throughout the protocol.
  • Cardiac function (LV pressure, wall thickening) and resistance artery responses to acetylcholine and endothelin-1 were evaluated.

Main Results:

  • Myocardial contractile function (LV pressure, wall thickening) was similarly depressed in vehicle- and cariporide-treated rats compared to controls.
  • Acetylcholine-induced relaxation was blunted in both vehicle and cariporide groups but was significantly greater in the cariporide group after 15 min of reperfusion.
  • Endothelin-1 contractile responses were similarly increased, while sodium nitroprusside relaxation was unchanged among groups.

Conclusions:

  • NHE(1) inhibition with cariporide attenuates ischemia-induced microvascular dysfunction in coronary resistance arteries.
  • NHE(1) inhibition does not improve myocardial contractile function in the area at risk following ischemia-reperfusion.
  • These findings suggest a specific role for NHE(1) in microvascular stunning, distinct from myocardial stunning.

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