[Pyridyl- and piperidyl-histamines (author's transl)]

Antihistaminic drugs modify casein-induced inflammation in the rat.

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Contractile properties of various histaprodifen derivatives in guinea pig isolated ileum and trachea.

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BF2.649 [1-{3-[3-(4-Chlorophenyl)propoxy]propyl}piperidine, hydrochloride], a nonimidazole inverse agonist/antagonist at the human histamine H3 receptor: Preclinical pharmacology.

The Journal of pharmacology and experimental therapeutics·2006

Piperidine-containing histamine H3 receptor antagonists of the carbamate series: the alkyl derivatives.

Die Pharmazie·2005

Search for histamine H3 receptor antagonists with combined inhibitory potency at Ntau-methyltransferase: ether derivatives.

Die Pharmazie·2005

Unexpected partial H1-receptor agonism of imidazole-type histamine H3-receptor antagonists lacking a basic side chain.

Inflammation research : official journal of the European Histamine Research Society ... [et al.]·2004

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Archiv der Pharmazie·2026

Design, Synthesis, and Biological Evaluation of Biphenylsulfonyl Indole-Based Thiosemicarbazones as Potential AChE and CA I-II Inhibitors.

Archiv der Pharmazie·2026

Targeting Human Protein Kinase CK2 by a Library of Indeno[1,2-b]Indoles: Contribution of Thermal Shift Assay to Pre-Screening and Co-Crystallization to Post-Screening.

Archiv der Pharmazie·2026

4-(5'-Dimethylamino)-Naphthalenesulfonyl-2(3H)-Benzoxazolone (W3D) Ameliorated COPD Lung Injury Through Regulating Macrophage Polarization Mediated by Glycolysis.

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Thiazole-Derived Dual EGFR/CDK-2 Inhibitors: Rational Design, Synthesis, In Vitro Anticancer Evaluation, Mechanistic Profiling, and Computational Binding Analysis.

Archiv der Pharmazie·2026

Anti-Inflammatory Effects of Ginsenosides: Molecular Mechanisms and Network Pharmacology Analysis.

The American journal of Chinese medicine·2026

Delicate Balance of Intra- and Inter-Molecular Entropic Effects in S-S Peptide Cyclization.

The journal of physical chemistry. A·2026

Distinct STRIPAK subunits drive conserved and subunit-specific signaling programs in Cryptococcus neoformans.

mBio·2026

Non-Destructive Analysis of Phenolic and Flavonoid Contents in Medicinal Plant Powders Using Hyperspectral Imaging and Variable Selection.

Analytical science advances·2026

Recent advances in multimodal foundation model-enabled peptide screening and optimization for smart biomaterials and functional tissue engineering.

Frontiers in bioengineering and biotechnology·2026

SP-3 Ameliorates Established Cyclophosphamide-Induced Liver Injury and Is Associated with PPAR-Related Transcriptional and Lipid-Metabolic Changes.

International journal of molecular sciences·2026

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[Pyridyl- and piperidyl-histamines (author's transl)]

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Antihistaminic drugs modify casein-induced inflammation in the rat.

Contractile properties of various histaprodifen derivatives in guinea pig isolated ileum and trachea.

BF2.649 [1-{3-[3-(4-Chlorophenyl)propoxy]propyl}piperidine, hydrochloride], a nonimidazole inverse agonist/antagonist at the human histamine H3 receptor: Preclinical pharmacology.

Piperidine-containing histamine H3 receptor antagonists of the carbamate series: the alkyl derivatives.

Search for histamine H3 receptor antagonists with combined inhibitory potency at Ntau-methyltransferase: ether derivatives.

Unexpected partial H1-receptor agonism of imidazole-type histamine H3-receptor antagonists lacking a basic side chain.

Breaking the Myb-KIX Alliance: Structure-Guided Discovery of Biaryl Hydroxy-Naphthamides as Disruptors of the c-Myb-CBP/p300 KIX Protein-Protein Interaction.

Discovery of VEGFR-2 Inhibitors From Leonurus japonicus via Integrated Genetic Authentication, Molecular Networking, and In Silico Analysis.

Design, Synthesis, and Biological Evaluation of Biphenylsulfonyl Indole-Based Thiosemicarbazones as Potential AChE and CA I-II Inhibitors.

Targeting Human Protein Kinase CK2 by a Library of Indeno[1,2-b]Indoles: Contribution of Thermal Shift Assay to Pre-Screening and Co-Crystallization to Post-Screening.

4-(5'-Dimethylamino)-Naphthalenesulfonyl-2(3H)-Benzoxazolone (W3D) Ameliorated COPD Lung Injury Through Regulating Macrophage Polarization Mediated by Glycolysis.

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Distinct STRIPAK subunits drive conserved and subunit-specific signaling programs in Cryptococcus neoformans.

Non-Destructive Analysis of Phenolic and Flavonoid Contents in Medicinal Plant Powders Using Hyperspectral Imaging and Variable Selection.

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[Pyridyl- and piperidyl-histamines (author's transl)]

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