Selective estrogen receptor modulators: tissue selectivity and differential uterine effects.

S L Silfen1, A V Ciaccia, H U Bryant

  • 1Eli Lilly and Company, Lilly Corporate Center, DC 2244, Indianapolis, IN, USA.

Summary

Selective estrogen receptor modulators (SERMs) offer tissue-specific effects, but their impact on the uterus varies. Raloxifene shows a favorable uterine safety profile compared to other SERMs.

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