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Small, low nanomolar, noncovalent thrombin inhibitors lacking a group to fill the 'distal binding pocket'

Philip E J Sanderson1, Kellie J Cutrona, Dona L Dyer

  • 1Department of Medicinal Chemistry, Merck Research Laboratories, West Point, PA 19486, USA. phil_sanderson@merck.com

Bioorganic & Medicinal Chemistry Letters
|December 17, 2002
PubMed

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