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Updated: Sep 27, 2026

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
10:33

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors

Published on: October 26, 2015

A substrate variant as a high-affinity, reversible inhibitor: insight from the X-ray structure of cilastatin bound to

Timothy P Smyth1, J Gerard Wall, Yasushi Nitanai

  • 1Department of Chemical and Environmental Sciences, Univeristy of Limerick, National Technological Park, County Limerick, Ireland. timothy.smyth@ul.ie

Bioorganic & Medicinal Chemistry
|March 5, 2003
PubMed

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