Na/H exchange isoform 1 is involved in mineralocorticoid/salt-induced cardiac injury

Genro Fujisawa1, Koji Okada, Shigeaki Muto

  • 1Division of Endocrinology and Metabolism, Department of Internal Medicine, Jichi Medical School, Minamikawachi, Tochigi, 329-0498 Japan. genrfjs@attglobal.net

Insights

The study shows that inhibiting Na/H exchange isoform 1 (NHE1) with cariporide prevents desoxycorticosterone acetate (DOCA)/salt-induced heart damage. This highlights NHE1

Area of Science:

  • Cardiovascular Research
  • Cellular Mechanisms
  • Pharmacology

Background:

  • Long-term desoxycorticosterone acetate (DOCA)/salt exposure causes cardiac fibrosis and hypertrophy via mineralocorticoid receptors (MRs).
  • The specific cellular pathways mediating these effects are not fully understood.

Purpose of the Study:

  • To investigate the role of Na/H exchange isoform 1 (NHE1) in DOCA/salt-induced cardiac damage.
  • To evaluate the efficacy of the NHE1 inhibitor cariporide and the MR antagonist spironolactone in preventing these changes.

Main Methods:

  • Uninephrectomized rats received DOCA/salt treatment for 8 days.
  • Groups were treated with spironolactone or cariporide.
  • Cardiac fibrosis, hypertrophy, and NHE1 protein expression were assessed.

Main Results:

  • Cariporide and spironolactone abolished DOCA/salt-induced perivascular collagen deposition.
  • Cariporide completely suppressed interstitial collagen deposition, while spironolactone partially suppressed it.
  • Cariporide completely inhibited DOCA/salt-induced cardiocyte hypertrophy and normalized increased NHE1 protein expression.

Conclusions:

  • Cardiac NHE1 plays a significant role in DOCA/salt-induced cardiac fibrosis and hypertrophy.
  • Cariporide effectively prevents DOCA/salt-induced cardiac injury, partly by inhibiting NHE1 activation.
  • DOCA/salt-induced cardiac injury mediated by MRs involves partial activation of NHE1.

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