Discovery of selective phosphonamide-based inhibitors of tumor necrosis factor-alpha converting enzyme (TACE)

Masaaki Sawa1, Kiriko Kurokawa, Yoshimasa Inoue

  • 1Department of Chemistry, R&D Laboratories, Nippon Organon K.K., 1-5-90, Tomobuchi-cho, Miyakojima-ku, 16, Osaka 534-00, Japan. masaaki-sawa@dainippon-pharm.co.jp

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