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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones

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Versatile and facile synthesis of diverse semisynthetic tetracycline derivatives via Pd-catalyzed reactions

Mark L Nelson1, Mohamed Y Ismail, Laura McIntyre

  • 1Paratek Pharmaceuticals, Inc., 75 Kneeland Street, Boston, Massachusetts 02111, USA. mnelson@paratekpharm.com

The Journal of Organic Chemistry
|July 19, 2003
PubMed

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