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Normal cardiac myosin ATPase and mechanics in pressure overload with digitalis treatment

Insights

Digitalis treatment prevents the decline in cardiac muscle myosin ATPase activity and contractile function caused by chronic pressure overload in cats. This indicates digitalis preserves heart function under stress.

Area of Science:

  • Cardiology
  • Biochemistry
  • Physiology

Background:

  • Chronic pressure overload impairs cardiac function by depressing myosin ATPase activity.
  • Digitalis administration can attenuate the decline in mechanical function during pressure overload.

Purpose of the Study:

  • To investigate the effect of digitalis on cardiac muscle myosin ATPase activity in cats with pressure overload.
  • To determine if digitalis maintains normal ATPase activity in parallel with mechanical function under chronic pressure overload.

Main Methods:

  • Four groups of cats were studied: controls, pressure-overload hypertrophy with or without failure (HF), digitalis-treated (D), and digitalis-treated with pressure overload (DHF).
  • Cardiac muscle myosin ATPase activity and papillary muscle isometric rate of force development were measured.

Main Results:

  • Myosin ATPase activity was significantly depressed in HF compared to controls (P < 0.05).
  • Digitalis treatment (D and DHF groups) did not significantly alter myosin ATPase activity compared to controls (P > 0.05).
  • Papillary muscle force development was depressed in HF but not in D or DHF groups compared to controls.

Conclusions:

  • The depression of cardiac myosin ATPase activity observed in heart failure due to pressure overload is prevented by concomitant digitalis administration.
  • Digitalis preserves both myosin ATPase activity and contractile function in the setting of chronic pressure overload.

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