Nuclear targeting of Akt enhances kinase activity and survival of cardiomyocytes

Isao Shiraishi1, Jaime Melendez, Youngkeun Ahn

  • 1The Children's Hospital Research Foundation, Division of Molecular Cardiovascular Biology; Cincinnati, Ohio, USA.

Circulation Research
|February 28, 2004
PubMed

Insights

Nuclear-targeted Akt inhibits cardiomyocyte apoptosis and protects the heart from injury without causing hypertrophy. This finding offers new therapeutic strategies for heart disease by targeting nuclear Akt signaling.

Area of Science:

  • Cardiology
  • Molecular Biology
  • Cell Biology

Background:

  • Heart failure involves cardiomyocyte death, reducing heart contractility.
  • Membrane-targeted Akt inhibits apoptosis, but nuclear Akt accumulation suggests nuclear targets.
  • Previous studies focused on membrane-bound Akt, overlooking its nuclear role.

Purpose of the Study:

  • To investigate the antiapoptotic effects of nuclear Akt accumulation.
  • To determine if nuclear Akt targeting prevents heart disease pathogenesis.
  • To explore therapeutic potential of nuclear-targeted Akt.

Main Methods:

  • Created and confirmed nuclear localization of an Akt construct using confocal microscopy.
  • Assessed cardiomyocyte apoptosis and remodeling in response to hypoxia.
  • Utilized transgenic models to evaluate nuclear Akt effects on heart function and gene expression.

Main Results:

  • Nuclear-targeted Akt effectively inhibited apoptosis, comparable to membrane-targeted Akt.
  • No hypertrophic remodeling or altered cardiomyocyte morphology was observed with nuclear Akt.
  • Transgenic hearts with nuclear Akt were protected from ischemia-reperfusion injury.
  • Gene array analysis revealed distinct transcriptional changes in nuclear Akt-expressing hearts.

Conclusions:

  • Targeting Akt to the nucleus inhibits apoptosis without inducing detrimental hypertrophic remodeling.
  • Nuclear Akt signaling represents a novel therapeutic avenue for heart disease.
  • This approach offers a way to prevent cell death in cardiac conditions.

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