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Updated: Aug 25, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Published on: August 16, 2018

Tricyclic pyridones as functionally selective human GABAA alpha 2/3 receptor-ion channel ligands

James Crawforth1, John R Atack, Susan M Cook

  • 1Department of Medicinal Chemistry, The Neuroscience Research Centre, Terlings Park, Eastwick Road, Harlow, Essex CM20 2QR, UK. james_crawforth@merck.com

Bioorganic & Medicinal Chemistry Letters
|March 18, 2004
PubMed

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