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Synthesis of a Borylated Ibuprofen Derivative Through Suzuki Cross-Coupling and Alkene Boracarboxylation Reactions
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A prodrug approach to COX-2 inhibitors with methylsulfone

Joo Hyun Moh1, Young Hoon Choi, Kyoung Min Lim

  • 1Drug Discovery, AmorePacific R&D Center, 314-1 Bora-ri, Giheung-eup, Yongin, Gyeonggi-do 449-729, Republic of Korea.

Bioorganic & Medicinal Chemistry Letters
|March 18, 2004
PubMed

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