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Updated: Aug 23, 2026

Genetically-encoded Molecular Probes to Study G Protein-coupled Receptors
Published on: September 13, 2013
Strategic Research Institute G-Protein-Coupled Receptors Drug Discovery World Summit
1Eli Lilly Research Laboratories, Neuroscience Division, Indianapolis, IN, USA. Felder@lilly.com
Abstract:
The Strategic Research Institute provided a well-organised 2-day summit that offered presentations and posters on new assay technology, structure-based small-molecule discovery and examples of clinical candidates targeted to G-protein-coupled receptor (GPCR) targets. A wide variety of topics were presented providing recent advances in GPCR target selection, bioassay-enabling technology and medicinal chemistry targeted to GPCR-relevant chemical libraries. GPCRs continue to be an attractive platform for drug discovery.
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