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Receptor Autoradiography Protocol for the Localized Visualization of Angiotensin II Receptors
Published on: June 7, 2016
Development of an efficient and selective radioligand for bradykinin B1 receptor occupancy studies
Dai-Shi Su1, M Kristine Markowitz, Kathy L Murphy
1Department of Medicinal Chemistry, Merck Research Laboratories, West Point, PA 19486, USA. daishi_su@merck.com
Bioorganic & Medicinal Chemistry Letters
|November 18, 2004
Abstract:
We have developed an efficient and selective radioligand, the [35S]-radiolabeled dihydroquinoxalinone derivative, 4, for an ex vivo receptor occupancy assay in transgenic rats over-expressing the human bradykinin B1 receptor.

