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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

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Synthesis and structure-activity relationships of novel histamine H1 antagonists: indolylpiperidinyl benzoic acid

Silvia Fonquerna1, Montse Miralpeix, Lluís Pagès

  • 1Almirall Prodesfarma S.A., Research Center, Cardener 68-74, 08024-Barcelona, Spain. sfonquerna@almirall.es

Journal of Medicinal Chemistry
|November 30, 2004
PubMed

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