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Identified a morpholinyl-4-piperidinylacetic acid derivative as a potent oral active VLA-4 antagonist

Jun Chiba1, Nobuo Machinaga, Tohru Takashi

  • 1Medicinal Chemistry Research Laboratory, Daiichi Pharmaceutical Co. Ltd, 16-13 Kitakasai 1-chome, Edogawa-ku, Tokyo 134-8630, Japan. chiba2mk@daiichipharm.co.jp

Bioorganic & Medicinal Chemistry Letters
|December 8, 2004
PubMed

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