Related Experiment Videos
Lunasin: a cancer-preventive soy peptide
1Department of Nutritional Sciences and Toxicology, University of California, 231 Morgan Hall, Berkeley, CA 94720-3104, USA. nitto@nature.berkeley.edu
Abstract:
Lunasin is a novel, cancer-preventive peptide whose efficacy against chemical carcinogens and oncogenes has been demonstrated in mammalian cells and in a skin cancer mouse model. Isolated and characterized in soy, lunasin peptide is also documented in barley. Lunasin is found in all of the genotypes analyzed from the US soy germ plasm collection and in commercially available soy proteins. Pilot studies show that lunasin is bioavailable in mice and rats when orally ingested, opening the way for dietary administration in cancer prevention studies. Lunasin internalizes into mammalian cells within minutes of exogenous application, and localizes in the nucleus after 18 hours. It inhibits acetylation of core histones in mammalian cells. In spite of its cancer-preventive properties, lunasin does not affect the growth rate of normal and established cancer cell lines. An epigenetic mechanism of action is proposed whereby lunasin selectively kills cells being transformed or newly transformed by binding to deacetylated core histones exposed by the transformation event, disrupting the dynamics of histone acetylation-deacetylation and leading to cell death.
Insights
Lunasin, a soy-derived peptide, shows cancer-preventive effects by selectively killing transformed cells through an epigenetic mechanism. This novel peptide is bioavailable and offers a promising avenue for dietary cancer prevention strategies.
Area of Science:
- Biochemistry
- Molecular Biology
- Oncology
Background:
- Lunasin is a unique, cancer-preventive peptide identified in soy and barley.
- It has demonstrated efficacy against chemical carcinogens and oncogenes in preclinical models.
- Lunasin is present in various soy germplasm and commercial soy protein products.
Purpose of the Study:
- To investigate the bioavailability and cellular mechanisms of lunasin.
- To explore lunasin's potential as a dietary agent for cancer prevention.
- To elucidate the epigenetic mechanism underlying lunasin's cancer-preventive properties.
Main Methods:
- Bioavailability studies in mice and rats following oral ingestion.
- Cellular uptake and localization experiments in mammalian cells.
- Analysis of histone acetylation inhibition and effects on cell lines.
Main Results:
- Lunasin is orally bioavailable in rodents.
- It rapidly internalizes into mammalian cells and localizes in the nucleus.
- Lunasin inhibits core histone acetylation without affecting normal or cancer cell growth.
- An epigenetic mechanism involving binding to deacetylated histones in transformed cells is proposed.
Conclusions:
- Lunasin exhibits cancer-preventive properties through a selective epigenetic mechanism.
- Its bioavailability supports its potential for dietary administration.
- Lunasin represents a promising candidate for novel cancer prevention strategies.
Related Concept Videos
Cancer Prevention
Some...
Cancer Prevention
Some...
Targeted Cancer Therapies
There are several types of targeted therapies against specific...
Loss of Tumor Suppressor Gene Functions
When the tumor suppressor genes develop mutations or are lost, cells start growing out of control, leading to cancer. However, a single functional copy of the tumor suppressor gene is enough for the cells to maintain their normal functions and cell...
Cancer-Critical Genes II: Tumor Suppressor Genes
When the function of certain critical genes, especially those involved in cell cycle regulation and cell growth signaling cascades, gets disrupted, it upsets the cell cycle progression. Such cells with unchecked cell cycles start proliferating uncontrollably and eventually develop into tumors.
Such genes that act...
Cancer-Critical Genes II: Tumor Suppressor Genes
When the function of certain critical genes, especially those involved in cell cycle regulation and cell growth signaling cascades, gets disrupted, it upsets the cell cycle progression. Such cells with unchecked cell cycles start proliferating uncontrollably and eventually develop into tumors.
Such genes that act...