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Updated: Feb 13, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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Allosteric modulation of dopamine receptors

John A Schetz1

  • 1Department of Pharmacology and Neuroscience, University of North Texas Health Sciences Center, 3500 Camp Bowie Blvd., Fort Worth, TX 76107, USA. jschetz@hsc.unt.edu

Mini Reviews in Medicinal Chemistry
|June 25, 2005
PubMed
Summary

Allosteric modulators precisely adjust dopamine receptor activity, offering new therapeutic strategies for diseases by fine-tuning responses to neurotransmitters and drugs.

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