Talnetant GlaxoSmithKline
1Menarini Ricerche SpA, Via Sette Santi 1, 50131, Firenze, Italy. sevangelista@menarini-recherche.it
Abstract:
Talnetant (SB-223412) is a selective, orally active NK3 antagonist based on 4-quinolinecarboxamide, and is under development by GlaxoSmithKline (formerly SmithKline Beecham) for the potential treatment of several disorders, including urinary incontinence, irritable bowel syndrome and schizophrenia. By November 2004, the compound had completed phase II trials.
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