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Preorganization of the hydroxyethylene dipeptide isostere: the preferred conformation in solution resembles the

Paloma Vidal1, David Timm, Howard Broughton

  • 1Discovery Chemistry Research and Technologies, Lilly Research Laboratories, Centro de Investigación Lilly, Avenida de la Industria 30, 28108 Alcobendas, Madrid, Spain.

Journal of Medicinal Chemistry
|November 24, 2005
PubMed

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