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Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
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Synthesis of deserpidine from reserpine

Greta Varchi1, Arturo Battaglia, Cristian Samorì

  • 1Istituto CNR per la Sintesi Organica e Fotoreattività ISOF, Area della Ricerca di Bologna, Via P., Gobetti 101, 40129 Bologna, Italy. G.Varchi@isof.cnr.it

Journal of Natural Products
|November 29, 2005
PubMed
Summary

Deserpidine, an antihypertensive drug, is synthesized from reserpine in six steps. This provides a viable alternative due to the limited natural availability of deserpidine.

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