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Updated: Aug 13, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
07:16

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

Clinical potential of GABAB receptor modulators

Jennifer Ong1, David I B Kerr

  • 1Department of Anaesthesia and Intensive Care, The University of Adelaide, Australia. jennifer.ong@adelaide.edu.au

CNS Drug Reviews
|January 4, 2006
PubMed
Summary

New phenylalkylamines act as positive allosteric modulators of GABAB receptors, offering a selective approach to drug discovery for neurological disorders without agonist side effects.

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