Discovery of nonpeptidic small-molecule AP-1 inhibitors: lead hopping based on a three-dimensional pharmacophore

Keiichi Tsuchida1, Hisaaki Chaki, Tadakazu Takakura

  • 1Discovery Laboratories, Toyama Chemical Co., Ltd., 4-1 Shimookui 2-chome, Toyama 930-8508, Japan. keiichi_tuchida@toyama-chemical.co.jp