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Stimulation of rabbit polymorphonuclear leukocyte locomotion by D-penicillamine

J G Elferink1, B M De Koster

  • 1Department of Medical Biochemistry, University of Leiden, The Netherlands.

Biochemical Pharmacology
|October 9, 1991
PubMed

Insights

Penicillamine enhances polymorphonuclear leukocyte (PMN) migration, acting as both a chemokinetic and chemotactic agent. This effect requires intact surface sulfhydryl groups and involves intracellular calcium, potentially linked to increased cGMP levels.

Area of Science:

  • Immunology
  • Cell Biology

Background:

  • Polymorphonuclear leukocytes (PMNs) are crucial immune cells involved in inflammatory responses.
  • Understanding factors that modulate PMN migration is vital for immune system research.

Purpose of the Study:

  • To investigate the effects of penicillamine on PMN migration and elucidate the underlying mechanisms.
  • To determine the role of cell surface sulfhydryl groups and intracellular calcium in penicillamine-induced PMN activation.

Main Methods:

  • Treatment of PMNs with penicillamine.
  • Assessing PMN chemotaxis and chemokinesis towards fMet-Leu-Phe.
  • Utilizing sulfhydryl reagents and calcium chelators to probe molecular mechanisms.
  • Measuring intracellular cyclic guanosine monophosphate (cGMP) levels.

Main Results:

  • Penicillamine significantly enhances PMN locomotion in the absence of chemoattractants, exhibiting both chemokinetic and chemotactic properties.
  • The activating effect of penicillamine is dependent on intact sulfhydryl groups on the PMN surface.
  • Intracellular calcium, but not extracellular calcium, plays a critical role in penicillamine-induced PMN migration enhancement.
  • Penicillamine treatment leads to an increase in intracellular cGMP levels within PMNs.

Conclusions:

  • Penicillamine modulates PMN migration through mechanisms involving cell surface sulfhydryl groups and intracellular calcium signaling.
  • The observed increase in cGMP levels may be associated with penicillamine's effects on PMN migration, although the direct relationship requires further investigation.

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