Related Experiment Video

Updated: Aug 9, 2026

Method for Identifying Small Molecule Inhibitors of the Protein-protein Interaction Between HCN1 and TRIP8b
10:20

Method for Identifying Small Molecule Inhibitors of the Protein-protein Interaction Between HCN1 and TRIP8b

Published on: November 11, 2016

Discovery of SB-705498: a potent, selective and orally bioavailable TRPV1 antagonist suitable for clinical

Harshad K Rami1, Mervyn Thompson, Geoffrey Stemp

  • 1Neurology and GI CEDD, New Frontiers Science Park, GlaxoSmithKline, Third Avenue, Harlow, Essex CM19 5AW, UK. Harshad.Rami@gsk.com

Bioorganic & Medicinal Chemistry Letters
|April 4, 2006
PubMed

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