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Updated: Aug 8, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

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CCK1 antagonists: are they ready for clinical use?

Shajan A S Peter1, Massimo D'Amato, Christoph Beglinger

  • 1Department of Gastroenterology, University Hospital, Basel, Switzerland.

Digestive Diseases (Basel, Switzerland)
|May 16, 2006
PubMed
Summary

Cholecystokinin (CCK) acts as both a hormone and neurotransmitter, regulating gastrointestinal functions and food intake. CCK1 antagonists show promise for treating GERD, IBS, pancreatitis, and other gastrointestinal disorders.

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