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Preparation of N-(2-alkoxyvinyl)sulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Preparation of N-(2-alkoxyvinyl)sulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines

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2,5-diketopiperazines as potent, selective, and orally bioavailable oxytocin antagonists. 3. Synthesis,

Alan D Borthwick1, Dave E Davies, Anne M Exall

  • 1Department of Medicinal Chemistry, Cardiovascular and Urogenital Centre of Excellence for Drug Discovery, Stevenage, UK. alan.d.borthwick@drugmoldesign.com

Journal of Medicinal Chemistry
|July 11, 2006
PubMed

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