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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Synthesis and identification of novel oxa-steroids as progesterone receptor antagonists

Fu-An Kang1, George Allan, Jihua Guan

  • 1Johnson and Johnson Pharmaceutical Research and Development, LLC, 665 Stockton Drive, Exton, PA 19341, USA. fkang@prdus.jnj.com

Bioorganic & Medicinal Chemistry Letters
|December 16, 2006
PubMed

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