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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Structure-activity relationships of novel piperazines as antagonists for the melanocortin-4 receptor

Dai Nozawa1, Taketoshi Okubo, Takaaki Ishii

  • 1Medicinal Research Laboratories, Taisho Pharmaceutical Co., Ltd, 1-403 Yoshino-cho, Kita-ku, Saitama, Saitama 331-9530, Japan. dai.nozawa@po.rd.taisho.co.jp

Bioorganic & Medicinal Chemistry
|January 20, 2007
PubMed

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