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Reverse Yeast Two-hybrid System to Identify Mammalian Nuclear Receptor Residues that Interact with Ligands and/or Antagonists
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Design, synthesis, and evaluation of non-steroidal farnesoid X receptor (FXR) antagonist

Masahiko Kainuma1, Makoto Makishima, Yuichi Hashimoto

  • 1Institute of Molecular and Cellular Biosciences, University of Tokyo, Yayoi, Bunkyo-ku, Tokyo 113-0032, Japan.

Bioorganic & Medicinal Chemistry
|February 13, 2007
PubMed

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