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Updated: Jul 14, 2026

Optimizing the Genetic Incorporation of Chemical Probes into GPCRs for Photo-crosslinking Mapping and Bioorthogonal Chemistry in Live Mammalian Cells
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Optimizing the Genetic Incorporation of Chemical Probes into GPCRs for Photo-crosslinking Mapping and Bioorthogonal Chemistry in Live Mammalian Cells

Published on: April 9, 2018

Bidirectional, iterative approach to the structural delineation of the functional "chemoprint" in GPR40 for agonist

Irina G Tikhonova1, Chi Shing Sum, Susanne Neumann

  • 1Laboratory of Biological Modeling, Clinical Endocrinology Branch, Chemical Biology Core Facility, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda, Maryland 20892, USA.

Journal of Medicinal Chemistry
|June 8, 2007
PubMed

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