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Updated: Jul 14, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Allosteric enhancers for A1 adenosine receptor.

Pier Giovanni Baraldi1, Maria Antonietta Iaconinoto, Allan R Moorman

  • 1Dipartimento di Scienze Farmaceutiche, Università di Ferrara, Ferrara, Italy. baraldi@unife.it

Mini Reviews in Medicinal Chemistry
|June 23, 2007
PubMed
Summary

Allosteric enhancers targeting the adenosine A(1) receptor show promise for treating cardiac arrhythmias and reducing fat breakdown. These compounds also offer potential as pain relievers and neuroprotective agents.

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