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A High-Throughput Enzyme-Coupled Activity Assay to Probe Small Molecule Interaction with the dNTPase SAMHD1
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A High-Throughput Enzyme-Coupled Activity Assay to Probe Small Molecule Interaction with the dNTPase SAMHD1

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Synthesis and biological activity of a gemcitabine phosphoramidate prodrug

Weidong Wu1, Jennifer Sigmond, Godefridus J Peters

  • 1Department of Medicinal Chemistry and Molecular Pharmacology and Cancer Center, Purdue University, West Lafayette, Indiana 47907, USA.

Journal of Medicinal Chemistry
|July 3, 2007
PubMed

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