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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Agonist potency at P2X7 receptors is modulated by structurally diverse lipids

A D Michel1, E Fonfria

  • 1Neurology & GI Centre of Excellence for Drug Discovery, GlaxoSmithKline Research & Development Limited, New Frontiers Science Park, Harlow, Essex, UK. adm7393@gsk.com

British Journal of Pharmacology
|August 19, 2007
PubMed
Abstract

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