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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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Parallel synthesis of 1,3-dihydro-1,4-benzodiazepine-2-ones employing catch and release

Line S Laustsen1, Christian K Sams

  • 1Medicinal Chemistry Research I, Chemical Research, Leo Pharma, Ballerup 2750, Denmark.

Journal of Combinatorial Chemistry
|October 6, 2007
PubMed

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