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Updated: Jul 10, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
07:16

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

GABA A/Bz receptor subtypes as targets for selective drugs

F Da Settimo1, S Taliani, M L Trincavelli

  • 1Dipartimento di Psichiatria, Neurobiologia, Farmacologia e Biotecnologie, Università di Pisa, Via Bonanno 6, 56126 Pisa, Italy.

Current Medicinal Chemistry
|November 6, 2007
PubMed
Summary

Targeting specific gamma-aminobutyric acid type A (GABA(A)) receptor subtypes with novel ligands offers potential for treating neurological disorders. Developing subtype-selective benzodiazepine site (BzR) ligands may lead to treatments with fewer side effects.

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