Cyclic guanidines as dual 5-HT5A/5-HT7 receptor ligands: optimising brain penetration

Jens-Uwe Peters1, Thomas Lübbers, Alexander Alanine

  • 1Discovery Chemistry, Pharma Division, F. Hoffmann-La Roche Ltd, CH-4070 Basel, Switzerland. jens-uwe.peters@roche.com

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