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Updated: Jul 9, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Heterotrimeric G protein activation by G-protein-coupled receptors

William M Oldham1, Heidi E Hamm

  • 1Department of Pharmacology, Vanderbilt University School of Medicine, 442 Robinson Research Building, 2222 Pierce Avenue, Nashville, TN 37232-6600, USA.

Nature Reviews. Molecular Cell Biology
|November 29, 2007
PubMed

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