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Updated: Jul 9, 2026

Detecting the Ligand-binding Domain Dimerization Activity of Estrogen Receptor Alpha Using the Mammalian Two-Hybrid Assay
09:07

Detecting the Ligand-binding Domain Dimerization Activity of Estrogen Receptor Alpha Using the Mammalian Two-Hybrid Assay

Published on: December 19, 2018

On the intractability of estrogen-related receptor alpha as a target for activation by small molecules

Stephen M Hyatt1, Elizabeth L Lockamy, Rebecca A Stein

  • 1Molecular Discovery Research Branch, GlaxoSmithKline, Research Triangle Park, NC 27709, USA.

Journal of Medicinal Chemistry
|December 7, 2007
PubMed

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