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Updated: Jul 9, 2026

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Quantitative Structure-Activity Relationship, Activity Prediction, and Molecular Dynamics of Non-nucleotide Reverse Transcriptase Inhibitors
Published on: May 9, 2025
Investigation of novel lipid-functionalized PNA monomers as potential HIV-1 non-nucleoside reverse transcriptase
Michael G Thomas1, Giovanni Maga, Jean-François Mouscadet
1Chemistry, School of Engineering & Physical Sciences, Heriot-Watt University, Edinburgh, United Kingdom.
Nucleosides, Nucleotides & Nucleic Acids
|December 7, 2007
Abstract:
A range of novel N-terminal lipid-functionalized peptide nucleic acid (PNA) monomers have been prepared and their abilities to inhibit HIV-1 reverse transcriptase and integrase have been examined.
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